Simona Rapposelli: шукати на сайті Z-Library

Sharifi-Rad, Javad, Rayess, Youssef El, Rizk, Alain Abi, Sadaka, Carmen, Zgheib, Raviella, Zam, Wissam, Sestito, Simona, Rapposelli, Simona, Neffe-SkociÅska, Katarzyna, ZieliÅska, Dorota, Salehi, Ba

Рік:

2006

Мова:

english

Файл:

PDF, 397 KB

english, 2006

Turmeric and Its Major Compound Curcumin on Health: Bioactive Effects and Safety Profiles for Food, Pharmaceutical, Biotechnological and Medicinal Applications

Журнал:

Frontiers in Pharmacology

Рік:

2020

Файл:

PDF, 1.63 MB

2020

Synthesis and 5-HT2A, 5-HT1A and α1-Binding Affinities of 2-[2-Hydroxy-3-(pyridin-3-yl-methyl)amino]-, 2-[2-Hydroxy-3-(2-pyridin-2-yl-ethyl)amino]- and 2-[2-Hydroxy-3-(4-N-methyl-piperazin-1-yl)-amino]propoxybenzaldehyde-O-(substituted) Benzyl Oximes

Elisabetta Orlandini, Simona Rapposelli, Susanna Nencetti, Gino Giannaccini, Laura Betti, Aldo Balsamo

Журнал:

Archiv der Pharmazie

Рік:

2007

Мова:

english

Файл:

PDF, 288 KB

english, 2007

Synthesis and Biological Evaluation of 2′-Oxo-2,3-dihydro-3′H- spiro[chromene-4,5′-[1,3]oxazolidin]-3′yl]acetic Acid Derivatives as Aldose Reductase Inhibitors

Simona Rapposelli, Federico Da Settimo, Maria Digiacomo, Concettina La Motta, Annalina Lapucci, Stefania Sartini, Michael Vanni

Журнал:

Archiv der Pharmazie

Рік:

2011

Мова:

english

Файл:

PDF, 254 KB

english, 2011

ChemInform Abstract: Synthesis and Inhibitory Activity Towards Human Leukocyte Elastase of New 7α-Methoxy and 7α-Chloro (2-Acyloxymethyl) Cephem Derivatives.

Aldo Balsamo, Giovanni Cercignani, Daniela Gentili, Annalina Lapucci, Marco Macchia, Elisabetta Orlandini, Simona Rapposelli, Armando Rossello

Журнал:

Aldo Balsamo, Simone Bertini, Giambattista Gervasi, Annalina Lapucci, Susanna Nencetti, Elisabetta Orlandini, Simona Rapposelli, Armando Rossello, Giulio Soldani

Рік:

2001

Файл:

PDF, 36 KB

2001

ChemInform Abstract: Enantiopure 3-(Arylmethylidene)aminoxy-2-methylpropionic Acids: Synthesis and Antiinflammatory Properties.

Журнал:

Рік:

2002

Файл:

PDF, 31 KB

2002

Conformationally Restrained Ceramide Analogues: Effects of Lipophilic Modifications on the Antiproliferative Activity.

Marco Macchia, Michela Antonello, Simone Bertini, Valeria Di Bussolo, Stefano Fogli, Elisa Giovannetti, Filippo Minutolo, Simona Rapposelli, Romano Danesi

Журнал:

Рік:

2003

Файл:

PDF, 14 KB

2003

Ceramide Analogues in Apoptosis: A New Strategy for Anticancer Drug Development

Marco Macchia, Simone Bertini, Stefano Fogli, Elisa Giovannetti, Filippo Minutolo, Simona Rapposelli, Romano Danesi

Журнал:

Рік:

2003

Файл:

PDF, 57 KB

2003

Synthesis and Prostaglandin Synthase Inhibitory Activity of New Aromatic O-Alkyloxime Ethers Substituted with Methylsulfonamido or Methylsulfonyl Groups on Their Aliphatic Portion.

Aldo Balsamo, Francesca Mancini, Claudio Milanese, Elisabetta Orlandini, Gabriella Ortore, Mario Pinza, Simona Rapposelli, Armando Rossello

Журнал:

Simona Rapposelli, Annalina Lapucci, Filippo Minutolo, Elisabetta Orlandini, Gabriella Ortore, Mario Pinza, Aldo Balsamo

Рік:

2004

Файл:

PDF, 124 KB

2004

Synthesis and COX-2 Inhibitory Properties of N-Phenyl- and N-Benzyl-Substituted Amides of 2-(4-Methylsulfonylphenyl)cyclopent-1-ene-1-carboxylic Acid and of Their Pyrazole, Thiophene and Isoxazole Analogues.

Журнал:

Filippo Minutolo, Michela Antonello, Simone Bertini, Giorgio Placanica, Simona Rapposelli, Kathryn E. Carlson, John A. Katzenellenbogen, Marco Macchia

Рік:

2004

Файл:

PDF, 132 KB

2004

Diaryl-Substituted Salicyl- and Anthranyl-ketoximes as Potential Estrogen Receptor Ligands.

Журнал:

Рік:

2004

Мова:

english

Файл:

PDF, 30 KB

english, 2004

Synthesis and Antimicrobial Activity of New 7β-(Benzo[a]dihydrocarbazolyloxyacetyl)-Substituted Cephalosporins.

Armando Rossello, Elisabetta Orlandini, Elisa Nuti, Simona Rapposelli, Marco Macchia, Enza Di Modugno, Aldo Balsamo

Журнал:

Рік:

2005

Файл:

PDF, 196 KB

2005

ChemInform Abstract: Synthesis and Biological Evaluation of 5-Membered Spiro Heterocycle-Benzopyran Derivatives Against Myocardial Ischemia.

Simona Rapposelli, Maria Cristina Breschi, Vincenzo Calderone, Maria Digiacomo, Alma Martelli, Lara Testai, Michael Vanni, Aldo Balsamo

Журнал:

Simona Rapposelli, Frederico Da Settimo, Maria Digiacomo, Concettina La Motta, Annalina Lapucci, Stefania Sartini, Michael Vanni

Рік:

2011

Файл:

PDF, 36 KB

2011

ChemInform Abstract: Synthesis and Biological Evaluation of [2′-Oxo-2,3-dihydro-3′H-spiro[chromene-4,5′- [1,3]oxazolidin]-3′yl]acetic Acid Derivatives as Aldose Reductase Inhibitors.

Журнал:

Рік:

2011

Файл:

PDF, 62 KB

2011

Synthesis of Stable Analogues of Geranylgeranyl Diphosphate Possessing a (Z,E,E)-Geranylgeranyl Side Chain, Docking Analysis, and Biological Assays for Prenyl Protein Transferase Inhibition

Filippo Minutolo, Simone Bertini, Laura Betti, Romano Danesi, Gianbattista Gervasi, Gino Giannaccini, Adriano Martinelli, Anna Maria Papini, Elisa Peroni, Giorgio Placanica, Simona Rapposelli, Tiziano

Журнал:

ChemMedChem

Рік:

2006

Мова:

english

Файл:

PDF, 398 KB

english, 2006

α-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors

Valentina Asso, Elisa Ghilardi, Simone Bertini, Maria Digiacomo, Carlotta Granchi, Filippo Minutolo, Simona Rapposelli, Andrea Bortolato, Stefano Moro, Marco Macchia

Журнал:

ChemMedChem

Рік:

2008

Мова:

english

Файл:

PDF, 355 KB

english, 2008

New N-arylsulfonyl-N-alkoxyaminoacetohydroxamic acids as selective inhibitors of gelatinase A (MMP-2)

Armando Rossello, Elisa Nuti, Elisabetta Orlandini, Paolo Carelli, Simona Rapposelli, Marco Macchia, Filippo Minutolo, Laura Carbonaro, Adriana Albini, Roberto Benelli, Giovanni Cercignani, Gillian Mu

Журнал:

Рік:

2004

Мова:

english

Файл:

PDF, 415 KB

english, 2004

Predictive models, based on classification algorithms, for compounds potentially active as mitochondrial ATP-sensitive potassium channel openers

Alessio Coi, Anna Maria Bianucci, Vincenzo Calderone, Lara Testai, Maria Digiacomo, Simona Rapposelli, Aldo Balsamo

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 381 KB

english, 2009

NO-glibenclamide derivatives: Prototypes of a new class of nitric oxide-releasing anti-diabetic drugs

Vincenzo Calderone, Simona Rapposelli, Alma Martelli, Maria Digiacomo, Lara Testai, Scilla Torri, Piero Marchetti, Maria C. Breschi, Aldo Balsamo

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2009

Мова:

english

Файл:

PDF, 355 KB

english, 2009

Stable analogues of geranylgeranyl diphosphate possessing improved geranylgeranyl versus farnesyl protein transferase inhibitory selectivity

Filippo Minutolo, Simone Bertini, Laura Betti, Romano Danesi, Gianbattista Gervasi, Gino Giannaccini, Chiara Papi, Giorgio Placanica, Silvia Barontini, Simona Rapposelli, Marco Macchia

Журнал:

Рік:

2003

Мова:

english

Файл:

PDF, 133 KB

english, 2003

A new development of matrix metalloproteinase inhibitors: twin hydroxamic acids as potent inhibitors of MMPs

Armando Rossello, Elisa Nuti, Maria Pia Catalani, Paolo Carelli, Elisabetta Orlandini, Simona Rapposelli, Tiziano Tuccinardi, Susan J. Atkinson, Gillian Murphy, Aldo Balsamo

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2005

Мова:

english

Файл:

PDF, 200 KB

english, 2005

Synthesis and biological evaluation of 5-membered spiro heterocycle-benzopyran derivatives against myocardial ischemia

Simona Rapposelli, Maria Cristina Breschi, Vincenzo Calderone, Maria Digiacomo, Alma Martelli, Lara Testai, Michael Vanni, Aldo Balsamo

Журнал:

Aldo Balsamo, Giovanni Cercignani, Daniela Gentili, Annalina Lapucci, Marco Macchia, Elisabetta Orlandini, Simona Rapposelli, Armando Rossello

Рік:

2011

Мова:

english

Файл:

PDF, 450 KB

english, 2011

Synthesis and inhibitory activity towards human leukocyte elastase of new 7α-methoxy and 7α-chloro (2-acyloxymethyl) cephem derivatives

Журнал:

Aldo Balsamo, Simone Bertini, Giambattista Gervasi, Annalina Lapucci, Susanna Nencetti, Elisabetta Orlandini, Simona Rapposelli, Armando Rossello, Giulio Soldani

Рік:

2001

Мова:

english

Файл:

PDF, 156 KB

english, 2001

Enantiopure 3-(arylmethylidene)aminoxy-2-methylpropionic acids: synthesis and antiinflammatory properties

Журнал:

Filippo Minutolo, Michela Antonello, Simone Bertini, Simona Rapposelli, Armando Rossello, Shubin Sheng, Kathryn E Carlson, John A Katzenellenbogen, Marco Macchia

Рік:

2001

Мова:

english

Файл:

PDF, 136 KB

english, 2001

Synthesis, binding affinity, and transcriptional activity of hydroxy- and methoxy-Substituted 3,4-Diarylsalicylaldoximes on estrogen receptors α and β

Журнал:

Рік:

2003

Мова:

english

Файл:

PDF, 308 KB

english, 2003

(E)-[2-(4-Methylsulphonylphenyl)-1-cyclopentenyl-1-methyliden](arylmethyloxy)amines. Methyleneaminoxymethyl (MAOM) analogues of diarylcyclopentenyl cyclooxygenase-2 inhibitors: synthesis and biological properties

Aldo Balsamo, Isabella Coletta, Paolo Domiano, Angelo Guglielmotti, Carla Landolfi, Francesca Mancini, Claudio Milanese, Elisabetta Orlandini, Simona Rapposelli, Mario Pinza, Bruno Macchia

Журнал:

Journal of Pharmacy and Pharmacology

Рік:

2002

Мова:

english

Файл:

PDF, 141 KB

english, 2002

Evaluation of the NO-releasing properties of NO-donor linkers

Vincenzo Calderone, Maria Digiacomo, Alma Martelli, Filippo Minutolo, Simona Rapposelli, Lara Testai, Aldo Balsamo

Журнал:

Рік:

2008

Мова:

english

Файл:

PDF, 234 KB

english, 2008

New NO-Releasing Pharmacodynamic Hybrids of Losartan and Its Active Metabolite: Design, Synthesis, and Biopharmacological Properties

Breschi, Maria C., Calderone, Vincenzo, Digiacomo, Maria, Macchia, Marco, Martelli, Alma, Martinotti, Enrica, Minutolo, Filippo, Rapposelli, Simona, Rossello, Armando, Testai, Lara

Журнал:

Simona Rapposelli, Annalina Lapucci, Filippo Minutolo, Elisabetta Orlandini, Gabriella Ortore, Mario Pinza, Aldo Balsamo

Рік:

2006

Мова:

english

Файл:

PDF, 222 KB

english, 2006

Anti-ischemic properties of a new spiro-cyclic benzopyran activator of the cardiac mito-KATP channel

Vincenzo Calderone, Lara Testai, Alma Martelli, Simona Rapposelli, Maria Digiacomo, Aldo Balsamo, Maria C. Breschi

Журнал:

Biochemical Pharmacology

Рік:

2010

Мова:

english

Файл:

PDF, 507 KB

english, 2010

Synthesis and COX-2 inhibitory properties of N-phenyl- and N-benzyl-substituted amides of 2-(4-methylsulfonylphenyl)cyclopent-1-ene-1-carboxylic acid and of their pyrazole, thiophene and isoxazole analogs

Журнал:

Рік:

2004

Мова:

english

Файл:

PDF, 263 KB

english, 2004

Synthesis of aniline-type analogues of farnesyl diphosphate and their biological assays for prenyl protein transferase inhibitory activity

Filippo Minutolo, Simone Bertini, Laura Betti, Valeria Di Bussolo, Gino Giannaccini, Giorgio Placanica, Simona Rapposelli, H.Peter Spielmann, Marco Macchia

Журнал:

Рік:

2003

Мова:

english

Файл:

PDF, 227 KB

english, 2003

Synthesis and antimicrobial activity of new 7β-(benzo[a]dihydrocarbazolyloxyacetyl)-substituted cephalosporins

Armando Rossello, Elisabetta Orlandini, Elisa Nuti, Simona Rapposelli, Marco Macchia, Enza Di Modugno, Aldo Balsamo

Журнал:

Filippo Minutolo, Michela Antonello, Simone Bertini, Giorgio Placanica, Simona Rapposelli, John A. Katzenellenbogen, Marco Macchia, Kathryn E. Carlson

Рік:

2004

Мова:

english

Файл:

PDF, 243 KB

english, 2004

Diaryl-substituted salicyl- and anthranyl-ketoximes as potential estrogen receptor ligands

Журнал:

Рік:

2004

Мова:

english

Файл:

PDF, 252 KB

english, 2004

Stable propylphosphonic acid analogues of geranylgeranyl diphosphate possessing inhibitory activity on geranylgeranyl protein transferase

Filippo Minutolo, Valentina Asso, Simone Bertini, Laura Betti, Gianbattista Gervasi, Elisa Ghilardi, Gino Giannaccini, Giorgio Placanica, Giovanni Prota, Simona Rapposelli, Marco Macchia

Журнал:

Рік:

2004

Мова:

english

Файл:

PDF, 194 KB

english, 2004

Phosphonomethylphosphorylmethyl(oxy)-analogues of geranylgeranyl diphosphate as stable and selective geranylgeranyl protein transferase inhibitors

Filippo Minutolo, Michela Antonello, Silvia Barontini, Simone Bertini, Laura Betti, Romano Danesi, Gianbattista Gervasi, Gino Giannaccini, Chiara Papi, Giorgio Placanica, Simona Rapposelli, Marco Macc

Журнал:

Рік:

2004

Мова:

english

Файл:

PDF, 209 KB

english, 2004

Conformationally restrained ceramide analogues: effects of lipophilic modifications on the antiproliferative activity

Marco Macchia, Michela Antonello, Simone Bertini, Valeria Di Bussolo, Stefano Fogli, Elisa Giovannetti, Filippo Minutolo, Simona Rapposelli, Romano Danesi

Журнал:

Рік:

2003

Мова:

english

Файл:

PDF, 150 KB

english, 2003

Ceramide analogues in apoptosis: a new strategy for anticancer drug development

Marco Macchia, Simone Bertini, Stefano Fogli, Elisa Giovannetti, Filippo Minutolo, Simona Rapposelli, Romano Danesi

Журнал:

Рік:

2003

Мова:

english

Файл:

PDF, 211 KB

english, 2003

Synthesis and prostaglandin synthase inhibitory activity of new aromatic O-alkyloxime ethers substituted with methylsulfonamido or methylsulfonyl groups on their aliphatic portion

Aldo Balsamo, Francesca Mancini, Claudio Milanese, Elisabetta Orlandini, Gabriella Ortore, Mario Pinza, Simona Rapposelli, Armando Rossello

Журнал:

Minutolo, Filippo, Antonello, Michela, Bertini, Simone, Ortore, Gabriella, Placanica, Giorgio, Rapposelli, Simona, Sheng, Shubin, Carlson, Kathryn E., Katzenellenbogen, Benita S., Katzenellenbogen, Jo

Рік:

2003

Мова:

english

Файл:

PDF, 320 KB

english, 2003

Novel Estrogen Receptor Ligands Based on an Anthranylaldoxime Structure: Role of the Phenol-Type Pseudocycle in the Binding Process

Журнал:

Grazia Chiellini, Simona Rapposelli, Jinge Zhu, Ilaria Massarelli, Marilena Saraceno, Anna Maria Bianucci, Lori A. Plum, Margaret Clagett-Dame, Hector F. DeLuca

Рік:

2003

Мова:

english

Файл:

PDF, 362 KB

english, 2003

Synthesis and biological activities of vitamin D-like inhibitors of CYP24 hydroxylase

Журнал:

Steroids

Рік:

2012

Мова:

english

Файл:

PDF, 1.36 MB

english, 2012

Design, synthesis and pharmacological evaluation of novel tacrine–caffeic acid hybrids as multi-targeted compounds against Alzheimer’s disease

Chao, Xiaojuan, He, Xixin, Yang, Yilin, Zhou, Xie, Jin, Minghua, Liu, Shu, Cheng, Zhiyi, Liu, Peiqing, Wang, Yuting, Yu, Jianchen, Tan, Yi, Huang, Yingjuan, Qin, Jian, Rapposelli, Simona, Pi, Rongbiao

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2012

Мова:

english

Файл:

PDF, 572 KB

english, 2012

Novel adenosine 5′-triphosphate-sensitive potassium channel ligands: a patent overview (2005 – 2010)

Rapposelli, Simona

Журнал:

Expert Opinion on Therapeutic Patents

Рік:

2011

Мова:

english

Файл:

PDF, 1.93 MB

english, 2011

Tacrine-6-Ferulic Acid, a Novel Multifunctional Dimer Against Alzheimer's Disease, Prevents Oxidative Stress-Induced Neuronal Death Through Activating Nrf2/ARE/HO-1 Pathway in HT22 Cells

Huang, Wen-Yong, Chao, Xiao-Juan, Ouyang, Ying, Liu, An-Min, He, Xi-Xin, Chen, Mei-Hui, Wang, Lan-Hua, Liu, Jun, Yu, Si-Wang, Rapposelli, Simona, Pi, Rong-Biao

Журнал:

CNS Neuroscience & Therapeutics

Рік:

2012

Мова:

english

Файл:

PDF, 150 KB

english, 2012

New Benzopyran-Based Openers of the Mitochondrial ATP-Sensitive Potassium Channel with Potent Anti-Ischemic Properties

Breschi, Maria C., Calderone, Vincenzo, Martelli, Alma, Minutolo, Filippo, Rapposelli, Simona, Testai, Lara, Tonelli, Federica, Balsamo, Aldo

Журнал:

Breschi, Maria C., Calderone, Vincenzo, Digiacomo, Maria, Manganaro, Mariaelisa, Martelli, Alma, Minutolo, Filippo, Rapposelli, Simona, Testai, Lara, Tonelli, Federica, Balsamo, Aldo

Рік:

2006

Мова:

english

Файл:

PDF, 115 KB

english, 2006

Spirocyclic Benzopyran-Based Derivatives as New Anti-ischemic Activators of Mitochondrial ATP-Sensitive Potassium Channel

Журнал:

Colabufo, Nicola Antonio, Berardi, Francesco, Perrone, Roberto, Rapposelli, Simona, Digiacomo, Maria, Vanni, Michael, Balsamo, Aldo

Рік:

2008

Мова:

english

Файл:

PDF, 203 KB

english, 2008

Sodium N -(Methylsulfonyl)- N -(4-nitro-2-phenoxyphenyl)sulfamate: A Water-Soluble Nimesulide Prodrug for Parenteral Use

Rapposelli, Simona, Digiacomo, Maria, Franchi, Silvia, Moretti, Sara, Pinza, Mario, Sacerdote, Paola, Balsamo, Aldo

Журнал:

Molecular Pharmaceutics

Рік:

2010

Мова:

english

Файл:

PDF, 246 KB

english, 2010

Synthesis and Biological Evaluation of (Hetero)Arylmethyloxy- and Arylmethylamine-phenyl Derivatives as Potent P-glycoprotein Modulating Agents

Журнал:

Rapposelli, Simona, Coi, Alessio, Imbriani, Marcello, Bianucci, Anna Maria

Рік:

2008

Мова:

english

Файл:

PDF, 255 KB

english, 2008

Development of Classification Models for Identifying “True” P-glycoprotein (P-gp) Inhibitors Through Inhibition, ATPase Activation and Monolayer Efflux Assays

Журнал:

International Journal of Molecular Sciences

Рік:

2012

Мова:

english

Файл:

PDF, 148 KB

english, 2012

NO-Sartans: A New Class of Pharmacodynamic Hybrids as Cardiovascular Drugs

Breschi, Maria C., Calderone, Vincenzo, Digiacomo, Maria, Martelli, Alma, Martinotti, Enrica, Minutolo, Filippo, Rapposelli, Simona, Balsamo, Aldo

Журнал:

Colabufo, Nicola Antonio, Berardi, Francesco, Perrone, Roberto, Rapposelli, Simona, Digiacomo, Maria, Vanni, Michael, Balsamo, Aldo

Рік:

2004

Мова:

english

Файл:

PDF, 129 KB

english, 2004

2-[(3-Methoxyphenylethyl)phenoxy]-Based ABCB1 Inhibitors: Effect of Different Basic Side-Chains on Their Biological Properties

Журнал: